Dermorphin

Product Overview

• Full Name: Dermorphin
• Amino Acid Sequence: Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NH₂
• Molecular Formula:C₄₀H₅₀N₈O₁₀
• Molecular Weight: ~802.87 g/mol
• CAS Number: 77614-16-5
• Core Mechanism

1. High selective μ-opioid receptor agonist with potent long-lasting analgesic effect.
2. Resist enzymatic degradation to extend pain relief duration.
3. Block central and spinal nociceptive signaling to ease acute and chronic pain.
4. Modulate inflammatory pain mediators to reduce nerve injury discomfort.

• Purity: ≥ 99% ( Endotoxin < 1 EU/mg)

Product Attributes

1. Ultra-potent long-duration pain relief

   Stronger analgesic activity than morphine, provides sustained relief for surgical and neuropathic pain.

2. Exclusive μ-opioid targeted ligand

   Minimal off-target binding to other opioid receptors, ideal for pain pathway research.

3. Mild gastrointestinal side effects compared to traditional opioids